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 4-methoxybenzo[d]thiazol-2-amine 4-methoxybenzo[d]thiazol-2(3H)-one 7-acetyl-4-(benzyloxy)-1,3-benzothiazol-2(3H)-one 4-(benzyloxy)-7-(bromoacetyl)-1,3-benzothiazol-2(3H)-one
 7-(2-azido-1-hydroxyethyl)-4-(benzyloxy)benzo[d]thiazol-2(3H)-one 7-[(1R)-2-azido-1-hydroxyethyl]-4-(benzyloxy)-1,3-benzothiazol-2(3H)-one (R)-7-(2-azido-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one 7-acetyl-4-methoxybenzo[d]thiazol-2(3H)-one
 7-(2-bromoacetyl)-4-hydroxybenzo[d]thiazol-2(3H)-one N-(2-chloro-4-formyl-5-methoxyphenyl)acrylamide 2-chloro-5-methoxyaniline 4-amino-5-chloro-2-methoxybenzaldehyde
 2-isocyanato-1,1’-biphenyl Tert-butyl 2-hydroxy-7-azaspiro[3.5]nonane-7-carboxylate 6-methoxyindoline 6-methoxyindoline-5-carbaldehyde
 Cis-tert-butyl 3,4-diazidopyrrolidine-1-carboxylate Cis-tert-butyl 3,4-dihydroxypyrrolidine-1-carboxylate GSK-961081; GSK-961081D; TD-5959; 961081; Batefenterol Succinate (R)-4-((3R,5R,8S,9S,10R,13R,14S,17R,E)-6-ethylidene-3-hydroxy-10,13-dimethyl-7-oxohexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanoic acid
 (R)-4-((3R,5S,8R,9S,10S,13R,14S,17R)-3-hydroxy-10,13-dimethyl-7-oxohexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanoic acid Obeticholic Acid;6-ECDCA; DSP-1747; INT-747 3-(5-methyl-1H-pyrrol-3-yl)propanoic acid 3-(4-(ethoxycarbonyl)-5-methyl-1H-pyrrol-3-yl)propanoic acid
 Afatinib;Gilotrif;BIBW 2992;Tovok 4-bromo-1-chloro-2-(4-ethoxybenzyl)benzene (2S,3R,4S,5S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6,6-bis(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol (2S,3R,4S,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol
 Ertugliflozin; PF 04971729;MK-8835 Sitagliptin phosphate;Januvia;Glactiv;ONO-5435; MK-0431; L-000224715 Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-3,4-dihydro-2H-pyran-3-yl)carbamate Tert-butyl ((1R,2S)-1-(2,5-difluorophenyl)-1-hydroxypent-4-yn-2-yl)carbamate
 Tert-butyl (1-(2,5-difluorophenyl)-1-oxopent-4-yn-2-yl)carbamate Tert-butyl (1-(methoxy(methyl)amino)-1-oxopent-4-yn-2-yl)carbamate 2-((tert-butoxycarbonyl)amino)pent-4-ynoic acid Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-5-hydroxytetrahydro-2H-pyran-3-yl)carbamate
 Tert-butyl ((2S,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2R,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2S,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole benzenesulfonate 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole Tert-butyl 6a-hydroxy-1,2,6,6a-tetrahydropyrrolo[3,4-c]pyrazole-5(4H)-carboxylate (Z)-tert-butyl 3-((dimethylamino)methylene)-4-oxopyrrolidine-1-carboxylate
 Tert-butyl 2-(methylsulfonyl)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole 4-methylbenzenesulfonate Tert-butyl 4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate (2S,3R,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
 AZD8186 PRT-060318;PRT318 Omarigliptin;MK-3102 (R)-2-(2-methoxyphenyl)-2-((tetrahydro-2H-pyran-4-yl)oxy)ethanol
 BGB-324 BAR 502 (S)-2-amino-3-(4-fluoro-1H-indol-3-yl)propanoic acid CMS-024; YSL; alpha-BCP[7-9];Tyroserleutide
 H3B-6527 BAR 501 AP-26113 , Brigatinib CCT251545
 RTA-402; NSC-713200; TP-155C; Methyl-CDDO; MethylCDDO;Bardoxolone methyl OTS-964 CCT251921 BLU-9931
 (R)-methyl 5-(6-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazol-1-yl)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-((5-((4-methylpiperazin-1-yl)methyl)-2-nitrophenyl)amino)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-amino-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-nitro-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate
 (S)-1-(2-(trifluoromethyl)phenyl)ethanol (S)-2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoic acid (S)-1-phenylethanamine (S)-2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoate 2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoic acid
 1-(3-fluoro-4-nitrobenzyl)-4-methylpiperazine 3-fluoro-4-nitrobenzaldehyde 3-fluoro-N-methoxy-N-methyl-4-nitrobenzamide methyl 3-hydroxy-5-nitrothiophene-2-carboxylate
 methyl 3-hydroxythiophene-2-carboxylate GSK-461364A PZM-21 BLU-554
 Nazartinib; EGF816; NVS-816 (S)-2-((2-(1-isopropyl-1H-1,2,4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)oxy)propanamide TEW-7197; NOV-1301; EW-7197 3-(N-(4-methyl-2-nitro-5-(pyridin-3-yl)phenyl)sulfamoyl)benzoic acid
 (2-((5-chloro-2-((2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)phenyl)dimethylphosphine oxide 1-(4-fluoro-1H-indol-3-yl)-N-((R)-1-phenylethyl)propan-2-amine 1-(4-fluoro-1H-indol-3-yl)propan-2-one (E)-4-fluoro-3-(2-nitroprop-1-en-1-yl)-1H-indole
 4-fluoro-1H-indole-3-carbaldehyde (S)-1-(4-fluoro-1H-indol-3-yl)propan-2-amine (R)-1-(4-fluoro-1H-indol-3-yl)propan-2-amine tert-butyl ((3S,4S)-4-azidotetrahydro-2H-pyran-3-yl)carbamate
 (3R,4R)-3-((tert-butoxycarbonyl)amino)tetrahydro-2H-pyran-4-yl methanesulfonate tert-butyl ((3R,4R)-4-hydroxytetrahydro-2H-pyran-3-yl)carbamate (3R,4R)-3-(((R)-1-phenylethyl)amino)tetrahydro-2H-pyran-4-ol 3,7-dioxabicyclo[4.1.0]heptane
 3,6-dihydro-2H-pyran (3S,4S)-4-azidotetrahydro-2H-pyran-3-amine hydrochloride CB-5083 N-(5-((4-(1H-indol-3-yl)pyrimidin-2-yl)amino)-2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methoxyphenyl)acrylamide
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