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 (3aS,3bR,7aS,8aS)-2,2,5,5-tetramethyltetrahydro-3aH-[1,3]dioxolo[4’,5’:4,5]furo[3,2-d][1,3]dioxine 1H-inden-1-yl)-2-methylpropane-2-sulfinamide AMG-232 ACP-103; BVF-048;Nuplazid;Pimavanserin Tartrate
 GS-7340-03; TAF; Tenofovir Alafenamide Fumarate BEC HCl 4-(2-(4-((5,5-dimethyl-1,4,2-dioxathiolan-3-yl)methoxy)phenyl)propan-2-yl)phenol (1S,2R)-2-tert-Butoxycarbonylamino-cyclohexylamine
 (5-methylpyridin-2-yl)methyl acetate 3-[1-(4-bromobenzyl)-3-tert-butylsulfanyl-5-hydroxy-1H-indol-2-yl]-2,2-dimethylpropionic acid ethyl ester 5-[4-(bromomethyl)phenyl]-2-(ethyloxy)pyridine hydrobromide (R)-N-((R)-4-cyano-2,3-dihydro-1H-inden-1-yl)-2-methylpropane-2-sulfinamide
 (S)-tert-butyl (4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)carbamate S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate (S)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile 6-benzyloxy-8-((R)-2-chloro-1-hydroxy-ethyl)-4H-benzo[1,4]-oxazin-3-one
 2-(3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)azetidin-3-yl)acetonitrile tert-butyl 3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-(cyanomethyl)azetidine-1-carboxylate 4-((1,5-dimethyl-1H-pyrazol-3-yl)amino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylic acid ethyl 4-amino-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylate
 ethyl 1-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrrole-2-carboxylate 8-chloroisoquinolin-3-amine (R)-1-(dimethylamino)propan-2-ol 6-chloro-5-iodopyrazin-2-amine
 3,8-dichloroisoquinoline (R)-5-amino-3-((1-(dimethylamino)propan-2-yl)oxy)pyrazine-2-carbonitrile 5-amino-3-chloropyrazine-2-carbonitrile 6-chloropyrazin-2-amine
 SAR-020106 2-fluoro-2-methylpropan-1-ol (S)-tert-butyl (1-(1H-indol-3-yl)-3-iodopropan-2-yl)carbamate 2-fluoro-2-methylpropyl trifluoromethanesulfonate
 ethyl 2-fluoro-2-methylpropanoate (S)-tert-butyl (1-hydroxy-3-(1H-indol-3-yl)propan-2-yl)carbamate (E)-methyl 3-(3,5-difluoro-4-formylphenyl)acrylate 2-(4-bromo-2-chlorophenyl)acetic acid
 4-(ethylaMino)-2-(Methylthio)pyriMidine-5-carbaldehyde (R)-tert-butyl 3-(6-amino-8-oxo-7H-purin-9(8H)-yl)piperidine-1-carboxylate (R)-tert-butyl 3-(6-(dibenzylamino)-8-oxo-7H-purin-9(8H)-yl)piperidine-1-carboxylate (R)-tert-butyl 3-((5-amino-6-(dibenzylamino)pyrimidin-4-yl)amino)piperidine-1-carboxylate
 GS-4059; ONO-4059 4-(3,4-dichloro-2-fluorophenylamino)-7-methoxyquinazolin-6-ol (2S,3R,4R,5S,6R)-2-(3-(benzo[b]thiophen-2-ylmethyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol (R)-2-((6-(3-aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl)-4-fluorobenzonitrile succinate
 2-((7-(3,4-dimethoxyphenyl)imidazo[1,2-c]pyrimidin-5-yl)amino)nicotinamide methyl 2-((7-(3,4-dimethoxyphenyl)imidazo[1,2-c]pyrimidin-5-yl)amino)nicotinate 5-chloro-7-(3,4-dimethoxyphenyl)imidazo[1,2-c]pyrimidine 7-(3,4-dimethoxyphenyl)imidazo[1,2-c]pyrimidin-5-ol
 7-(3,4-dimethoxyphenyl)-5-(ethylthio)imidazo[1,2-c]pyrimidine 6-(3,4-dimethoxyphenyl)-2-(ethylthio)pyrimidin-4-amine 4-amino-6-(3,4-dimethoxyphenyl)pyrimidine-2(1H)-thione (Z)-3-amino-3-(3,4-dimethoxyphenyl)acrylonitrile
 BAY-61-3606 5-(1-benzyl-1H-indazol-3-yl)furan-2-carbaldehyde 1-benzyl-3-(furan-2-yl)-1H-indazole 1-benzyl-3-iodo-1H-indazole
 3-iodo-1H-indazole YC-1 (2S,3S,4R,5R,6S)-5-(benzyloxy)-6-((5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-4-oxo-4H-chromen-3-yl)oxy)-2-methyltetrahydro-2H-pyran-3,4-diyl diacetate (2S,3S,4R,5R,6S)-5-(benzyloxy)-6-bromo-2-methyltetrahydro-2H-pyran-3,4-diyl diacetate
 (2S,3S,4R,5R,6S)-5-(benzyloxy)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4-diyl diacetate (2S,3R,4R,5R,6S)-5-(benzyloxy)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4-diol (4aS,5S,7S,8R,8aR)-8-(benzyloxy)-2,3-dimethoxy-2,3,5-trimethyl-7-(phenylthio)hexahydro-2H-pyrano[3,4-b][1,4]dioxine (4aS,5S,7S,8R,8aS)-2,3-dimethoxy-2,3,5-trimethyl-7-(phenylthio)hexahydro-2H-pyrano[3,4-b][1,4]dioxin-8-ol
 (2S,3R,4R,5R,6S)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4,5-triol (2S,3S,4R,5R,6S)-2-methyl-6-(phenylthio)tetrahydro-2H-pyran-3,4,5-triyl triacetate (2S,3R,4R,5S,6S)-6-methyltetrahydro-2H-pyran-2,3,4,5-tetrayl tetraacetate 5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-3-hydroxy-4H-chromen-4-one
 5,7-bis(benzyloxy)-2-(4-(benzyloxy)phenyl)-4H-chromen-4-one (E)-3-(4-(benzyloxy)phenyl)-1-(2,4-bis(benzyloxy)-6-hydroxyphenyl)prop-2-en-1-one SL-0101 5-cyano-2’-(piperazin-1-yl)-N-(3-(pyrrolidin-1-yl)propyl)-[1,1’-biphenyl]-3-carboxamide
 tert-butyl 4-(3’-cyano-5’-((3-(pyrrolidin-1-yl)propyl)carbamoyl)-[1,1’-biphenyl]-2-yl)piperazine-1-carboxylate 2’-bromo-5-cyano-N-(3-(pyrrolidin-1-yl)propyl)-[1,1’-biphenyl]-3-carboxamide LLY-507 2,2-dimethyl-4-((4-(2-(4-(oxiran-2-ylmethoxy)phenyl)propan-2-yl)phenoxy)methyl)-1,3-dioxolane
 EPI-001 ETC-1002 (ESP 55016),Bempedoic Acid 2-(3-bromophenyl)-N-((3’-(methylsulfonyl)-[1,1’-biphenyl]-4-yl)methyl)ethanamine 3’-(methylsulfonyl)-[1,1’-biphenyl]-4-carboxylic acid
 SR9243 N-(2-oxoindolin-5-yl)-3-(piperidin-1-yl)propanamide 5-aminoindolin-2-one DEL-22379,HY-18932
 MCB-613 (R)-tert-butyl 3-((6-(dibenzylamino)-5-nitropyrimidin-4-yl)amino)piperidine-1-carboxylate N,N-dibenzyl-6-chloro-5-nitropyrimidin-4-amine ethyl 4-((1,5-dimethyl-1H-pyrazol-3-yl)amino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylate
 3-iodo-1,5-dimethyl-1H-pyrazole 1,5-dimethyl-1H-pyrazol-3-amine ethyl 4-(4-cyano-1-methyl-1H-imidazol-5-yl)-1-ethyl-1H-pyrrole-2-carboxylate 5-bromo-1-methyl-1H-imidazole-4-carbonitrile
 1-methyl-1H-imidazole-4-carbonitrile (E)-3-(pyrrolidin-1-yl)-2-((E)-(pyrrolidin-1-ylmethylene)amino)acrylonitrile ethyl 4-bromo-1-ethyl-1H-pyrrole-2-carboxylate ethyl 4-bromo-1H-pyrrole-2-carboxylate
 1-(4-bromo-1H-pyrrol-2-yl)-2,2,2-trichloroethanone BMS-911543 1-(6-methylpyridin-2-yl)-2-(1,5-naphthyridin-2-yl)ethanone 2-methyl-1,5-naphthyridine
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