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 Alk5i 1-(((S)-3-(diethylamino)-2-hydroxypropyl)amino)-4-(((S)-oxiran-2-ylmethyl)amino)anthracene-9,10-dione sodium 4-methylbenzenesulfonate (E)-3-tosylacrylonitrile
 (Z)-3-(((4-((dimethylamino)methyl)phenyl)amino)(phenyl)methylene)-6-iodoindolin-2-one (E)-6-iodo-3-(phenyl((trimethylsilyl)oxy)methylene)-2-((trimethylsilyl)oxy)-3H-indole (S)-tert-butyl 4-((((9H-fluoren-9-yl)methoxy)carbonyl)amino)-5-(((S)-1-(allyloxy)-3-methyl-1-oxobutan-2-yl)amino)-5-oxopentanoate (S)-allyl 2-amino-3-methylbutanoate
 Ac-DEVD-CHO (E)-methyl 4-(3-(dimethylamino)-2-methylacryloyl)-1-tosyl-1H-pyrrole-2-carboxylate methyl 4-propionyl-1-tosyl-1H-pyrrole-2-carboxylate methyl 4-propionyl-1H-pyrrole-2-carboxylate
 1-(5-(2,2,2-trichloroacetyl)-1H-pyrrol-3-yl)propan-1-one VX-11e 1-(3-fluoro-2-(trifluoromethyl)isonicotinoyl)piperidin-4-one piperidin-4-one hydrochloride
 tert-butyl 3-(cyanomethyl)-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)azetidine-1-carboxylate tert-butyl 3-(cyanomethylene)azetidine-1-carboxylate tert-butyl 3-oxoazetidine-1-carboxylate tert-butyl 3-hydroxyazetidine-1-carboxylate
 INCB39110 (1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl)boronic acid 1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazole 8-ethyl-4-methyl-2-(methylthio)-6-(1H-pyrazol-5-yl)pyrido[2,3-d]pyrimidin-7(8H)-one
 8-ethyl-4-methyl-2-(methylthio)pyrido[2,3-d]pyrimidin-7(8H)-one (E)-ethyl 3-(4-(ethylamino)-6-methyl-2-(methylthio)pyrimidin-5-yl)acrylate N-ethyl-5-iodo-6-methyl-2-(methylthio)pyrimidin-4-amine N-ethyl-6-methyl-2-(methylthio)pyrimidin-4-amine
 4-chloro-6-methyl-2-(methylthio)pyrimidine 6-methyl-2-(methylthio)pyrimidin-4(3H)-one Voxtalisib (XL765, SAR245409) thiazol-5-ylboronic acid
 2-(trimethylsilyl)thiazole 6-(4-bromo-2-chlorophenyl)-8-ethyl-2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one 6-(4-bromo-2-chlorophenyl)-2-chloro-8-ethylpyrido[2,3-d]pyrimidin-7(8H)-one methyl 2-(4-bromo-2-chlorophenyl)acetate
 2-(4-bromo-2-chlorophenyl)acetonitrile 4-bromo-1-(bromomethyl)-2-chlorobenzene 2-chloro-4-(ethylamino)pyrimidine-5-carbaldehyde (2-chloro-4-(ethylamino)pyrimidin-5-yl)methanol
 ethyl 2-chloro-4-(ethylamino)pyrimidine-5-carboxylate FRAX597 ethyl 3-(3-(tert-butylthio)-1-(4-(6-ethoxypyridin-3-yl)benzyl)-5-((5-methylpyridin-2-yl)methoxy)-1H-indol-2-yl)-2,2-dimethylpropanoate 2-ethoxy-5-(4-((1-(4-((5-methylpyridin-2-yl)methoxy)phenyl)hydrazinyl)methyl)phenyl)pyridine
 4-((5-methylpyridin-2-yl)methoxy)aniline 5-(4-(bromomethyl)phenyl)-2-ethoxypyridine (4-(6-ethoxypyridin-3-yl)phenyl)methanol GSK2190915 (AM803)
 2,3,5-trifluoro-N-(3-fluoro-4-iodophenyl)-6-nitroaniline (S)-1-((2,2-dimethyl-1,3-dioxolan-4-yl)methyl)cyclopropane-1-sulfonyl chloride (S)-butyl 1-(3-((tert-butyldimethylsilyl)oxy)-2-hydroxypropyl)cyclopropane-1-sulfonate O-(2-(vinyloxy)ethyl)hydroxylamine
 2-(2-(vinyloxy)ethoxy)isoindoline-1,3-dione 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-N-(2-(vinyloxy)ethoxy)-1H-benzo[d]imidazole-6-carboxamide 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-1H-benzo[d]imidazole-6-carboxylic acid methyl 6-((4-bromo-2-fluorophenyl)amino)-7-fluoro-1H-benzo[d]imidazole-5-carboxylate
 methyl 4-amino-2-((4-bromo-2-fluorophenyl)amino)-3-fluoro-5-nitrobenzoate MEK162 5-((2S,3S,4R)-3,4-diaminotetrahydrothiophen-2-yl)pentanoic acid 5-((3aS,4S,6aR)-1,3-dibenzyl-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoic acid
 ethyl 5-((3aS,4S,6aR)-1,3-dibenzyl-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoate ethyl 5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoate (2-bromo-1,4-phenylene)dimethanol dimethyl 2-bromoterephthalate
 2-bromo-1,4-bis(((2-methoxypropan-2-yl)oxy)methyl)benzene (S)-methyl 2-((tert-butoxycarbonyl)amino)-3-(4-cyano-2,6-dimethylphenyl)propanoate (R)-(2-((tert-butoxycarbonyl)amino)-3-methoxy-3-oxopropyl)zinc(II) iodide (S)-2-((tert-butoxycarbonyl)amino)-3-(4-carbamoyl-2,6-dimethylphenyl)propanoic acid
 (S)-1-bromo-3-(1-(hexyloxy)ethyl)-2-methoxybenzene (S)-1-(3-bromo-2-methoxyphenyl)ethanol 1-(3-bromo-2-methoxyphenyl)ethanone 1-(3-bromo-2-methoxyphenyl)ethanol
 (S)-2-chloro-1-(3-(1-(hexyloxy)ethyl)-2-methoxyphenyl)ethanone 3,5-dichloro-4-formylbenzoic acid (E)-3,5-dichloro-4-(3-methoxy-2-methyl-3-oxoprop-1-en-1-yl)benzoic acid (R)-2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid
 (S)-2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid 2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid 8-cyclopentyl-5-methyl-2-(methylthio)pyrido[2,3-d]pyrimidin-7(8H)-one 1-(4-(cyclopentylamino)-2-(methylthio)pyrimidin-5-yl)ethanol
 4-(cyclopentylamino)-2-(methylthio)pyrimidine-5-carbaldehyde (4-(cyclopentylamino)-2-(methylthio)pyrimidin-5-yl)methanol ethyl 4-(cyclopentylamino)-2-(methylthio)pyrimidine-5-carboxylate 6-bromo-8-cyclopentyl-5-methyl-2-(methylsulfinyl)pyrido[2,3-d]pyrimidin-7(8H)-one
 (R)-8-(2-azido-1-((tert-butyldimethylsilyl)oxy)ethyl)-5-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one tert-butyl 2-(spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-ylidene)acetate spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-one 3-methylenespiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolane]
 spiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-one (2S)-2-bromospiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-one (1R,2S,3S,5R)-2-bromospiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-ol tert-butyl 2-((6S)-6-(nitromethyl)spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-yl)acetate
 4-(2-cyclopropylethyl)-3-hydroxyhept-6-enoic acid ethyl 4-(2-cyclopropylethyl)-3-hydroxyhept-6-enoate ethyl 4-(2-cyclopropylethyl)-3-oxohept-6-enoate ethyl 6-cyclopropyl-3-oxohexanoate
 (2-bromoethyl)cyclopropane (1R,5S)-3-(2-cyclopropylethyl)bicyclo[3.2.0]hept-3-en-6-one (S)-S-isopropyl 2-((tert-butoxycarbonyl)amino)propanethioate tert-butyl 2-((1S,5R,6R)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetate
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