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 1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazole 8-ethyl-4-methyl-2-(methylthio)-6-(1H-pyrazol-5-yl)pyrido[2,3-d]pyrimidin-7(8H)-one 8-ethyl-4-methyl-2-(methylthio)pyrido[2,3-d]pyrimidin-7(8H)-one (E)-ethyl 3-(4-(ethylamino)-6-methyl-2-(methylthio)pyrimidin-5-yl)acrylate
 N-ethyl-5-iodo-6-methyl-2-(methylthio)pyrimidin-4-amine N-ethyl-6-methyl-2-(methylthio)pyrimidin-4-amine 4-chloro-6-methyl-2-(methylthio)pyrimidine 6-methyl-2-(methylthio)pyrimidin-4(3H)-one
 Voxtalisib (XL765, SAR245409) thiazol-5-ylboronic acid 2-(trimethylsilyl)thiazole 6-(4-bromo-2-chlorophenyl)-8-ethyl-2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one
 6-(4-bromo-2-chlorophenyl)-2-chloro-8-ethylpyrido[2,3-d]pyrimidin-7(8H)-one methyl 2-(4-bromo-2-chlorophenyl)acetate 2-(4-bromo-2-chlorophenyl)acetonitrile 4-bromo-1-(bromomethyl)-2-chlorobenzene
 2-chloro-4-(ethylamino)pyrimidine-5-carbaldehyde (2-chloro-4-(ethylamino)pyrimidin-5-yl)methanol ethyl 2-chloro-4-(ethylamino)pyrimidine-5-carboxylate FRAX597
 ethyl 3-(3-(tert-butylthio)-1-(4-(6-ethoxypyridin-3-yl)benzyl)-5-((5-methylpyridin-2-yl)methoxy)-1H-indol-2-yl)-2,2-dimethylpropanoate 2-ethoxy-5-(4-((1-(4-((5-methylpyridin-2-yl)methoxy)phenyl)hydrazinyl)methyl)phenyl)pyridine 4-((5-methylpyridin-2-yl)methoxy)aniline 5-(4-(bromomethyl)phenyl)-2-ethoxypyridine
 (4-(6-ethoxypyridin-3-yl)phenyl)methanol GSK2190915 (AM803) 2,3,5-trifluoro-N-(3-fluoro-4-iodophenyl)-6-nitroaniline (S)-1-((2,2-dimethyl-1,3-dioxolan-4-yl)methyl)cyclopropane-1-sulfonyl chloride
 (S)-butyl 1-(3-((tert-butyldimethylsilyl)oxy)-2-hydroxypropyl)cyclopropane-1-sulfonate O-(2-(vinyloxy)ethyl)hydroxylamine 2-(2-(vinyloxy)ethoxy)isoindoline-1,3-dione 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-N-(2-(vinyloxy)ethoxy)-1H-benzo[d]imidazole-6-carboxamide
 5-((4-bromo-2-fluorophenyl)amino)-4-fluoro-1-methyl-1H-benzo[d]imidazole-6-carboxylic acid methyl 6-((4-bromo-2-fluorophenyl)amino)-7-fluoro-1H-benzo[d]imidazole-5-carboxylate methyl 4-amino-2-((4-bromo-2-fluorophenyl)amino)-3-fluoro-5-nitrobenzoate MEK162
 5-((2S,3S,4R)-3,4-diaminotetrahydrothiophen-2-yl)pentanoic acid 5-((3aS,4S,6aR)-1,3-dibenzyl-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoic acid ethyl 5-((3aS,4S,6aR)-1,3-dibenzyl-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoate ethyl 5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanoate
 (2-bromo-1,4-phenylene)dimethanol dimethyl 2-bromoterephthalate 2-bromo-1,4-bis(((2-methoxypropan-2-yl)oxy)methyl)benzene (S)-methyl 2-((tert-butoxycarbonyl)amino)-3-(4-cyano-2,6-dimethylphenyl)propanoate
 (R)-(2-((tert-butoxycarbonyl)amino)-3-methoxy-3-oxopropyl)zinc(II) iodide (S)-2-((tert-butoxycarbonyl)amino)-3-(4-carbamoyl-2,6-dimethylphenyl)propanoic acid (S)-1-bromo-3-(1-(hexyloxy)ethyl)-2-methoxybenzene (S)-1-(3-bromo-2-methoxyphenyl)ethanol
 1-(3-bromo-2-methoxyphenyl)ethanone 1-(3-bromo-2-methoxyphenyl)ethanol (S)-2-chloro-1-(3-(1-(hexyloxy)ethyl)-2-methoxyphenyl)ethanone 3,5-dichloro-4-formylbenzoic acid
 (E)-3,5-dichloro-4-(3-methoxy-2-methyl-3-oxoprop-1-en-1-yl)benzoic acid (R)-2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid (S)-2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid 2-(2-(benzyloxy)-3-isopropylphenyl)propanoic acid
 8-cyclopentyl-5-methyl-2-(methylthio)pyrido[2,3-d]pyrimidin-7(8H)-one 1-(4-(cyclopentylamino)-2-(methylthio)pyrimidin-5-yl)ethanol 4-(cyclopentylamino)-2-(methylthio)pyrimidine-5-carbaldehyde (4-(cyclopentylamino)-2-(methylthio)pyrimidin-5-yl)methanol
 ethyl 4-(cyclopentylamino)-2-(methylthio)pyrimidine-5-carboxylate 6-bromo-8-cyclopentyl-5-methyl-2-(methylsulfinyl)pyrido[2,3-d]pyrimidin-7(8H)-one (R)-8-(2-azido-1-((tert-butyldimethylsilyl)oxy)ethyl)-5-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one tert-butyl 2-(spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-ylidene)acetate
 spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-one 3-methylenespiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolane] spiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-one (2S)-2-bromospiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-one
 (1R,2S,3S,5R)-2-bromospiro[bicyclo[3.2.0]heptane-6,2’-[1,3]dioxolan]-3-ol tert-butyl 2-((6S)-6-(nitromethyl)spiro[bicyclo[3.2.0]heptane-3,1’-cyclopropan]-6-yl)acetate 4-(2-cyclopropylethyl)-3-hydroxyhept-6-enoic acid ethyl 4-(2-cyclopropylethyl)-3-hydroxyhept-6-enoate
 ethyl 4-(2-cyclopropylethyl)-3-oxohept-6-enoate ethyl 6-cyclopropyl-3-oxohexanoate (2-bromoethyl)cyclopropane (1R,5S)-3-(2-cyclopropylethyl)bicyclo[3.2.0]hept-3-en-6-one
 (S)-S-isopropyl 2-((tert-butoxycarbonyl)amino)propanethioate tert-butyl 2-((1S,5R,6R)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetate ethyl 2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetate ethyl 2-((1R,5S,6S)-3-ethyl-6-(nitromethyl)bicyclo[3.2.0]hept-3-en-6-yl)acetate
 (E)-ethyl 2-((1R,5S)-3-ethylbicyclo[3.2.0]hept-3-en-6-ylidene)acetate 3-ethylbicyclo[3.2.0]hept-3-en-6-one 4-ethyl-3-hydroxyhept-6-enoic acid ethyl 4-ethyl-3-hydroxyhept-6-enoate
 ethyl 4-ethyl-3-oxohept-6-enoate (cis)-tert-butyl 3-fluoro-4-hydroxypiperidine-1-carboxylate methyl 5-(N-methylacrylamido)pentanoate methyl 5-(methylamino)pentanoate
 5-(methylamino)pentanoic acid S-isopropyl 2-((tert-butoxycarbonyl)amino)-2-methylpropanethioate 4-amino-5-ethynyl-2-methoxybenzaldehyde spiro[[1,3]dioxolane-2,4’-tricyclo[5.2.0.02,5]nonane]
 spiro[[1,3]dioxolane-2,4’-tricyclo[5.2.0.02,5]nonan]-8’-one 9’,9’-dichlorospiro[[1,3]dioxolane-2,4’-tricyclo[5.2.0.02,5]nonan]-8’-one tricyclo[5.2.0.02,5]nonan-4-one 2,5-dimethoxy-2-methyl-2,5-dihydrofuran
 tert-butyl 2-(([1,1’-biphenyl]-2-ylcarbamoyl)oxy)-7azaspiro[3.5]nonane-7-carboxylate bicyclo[3.2.0]hept-3-en-6-one 3-hydroxyhept-6-enoic acid ethyl 3-oxohept-6-enoate
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