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 Ethyl 3-(cyanomethylene)cyclobutanecarboxylate Methyl 3-(cyanomethylene)cyclobutanecarboxylate Methyl 2-amino-5-propyl-1,3-thiazole-4-carboxylate t-Butyl 2-bromoisovalerate
 Methyl 2-methyl-3-oxopentanoate 4-Bromo-2-methoxy-6-methylaniline Ethyl 2-aminooxazole-4-carboxylate 3-Amino-6-methoxypyridazine
 2-Aminothiazol-4-acetic acid N-Boc-1,4-cyclohexanediamine 7-Bromo-2,3-dihydro-isoindol-1-one 2,4-Dichloropyrrolo[1,2-f][1,2,4]triazine
 2-Bromo-4-amino-5-methylpyridine Methyl 4-amino-5-methylthiophene-3-carboxylate tert-Butyl 3-butenoate Cyclobutane-1,1-diyldimethanol
 Benzyl 3-aminocyclobutylcarbamate 5-Ethoxy-2-ethoxycarbonyloxazole Methyl 2-(2-oxocyclohexyl)acetate 1-Methylcyclobutanol
 Ethyl 4-(dimethylamino)-2-oxobut-3-enoate 5-Amino-3-methyl-1H-thieno[3,2-c]pyrazole-6-carbonitrile 2,4-Dihydroxy-8-methylquinazoline 1-Methylpiperazin-2-one
 Ethyl 2-(3-oxocyclohexyl)acetate 3,4-Dichloropyridine-5-carboxylic acid 2-Methyl-4-phenylpyrimidine 2-(Chloromethyl)-4-phenylpyrimidine
 4-Chloro-6-methoxy-2-methylpyrimidine 1-Aminomethylcycloheptanol Ethyl 3-cyclopropyl-2,2-difluoropropanoate 4,6-Diamino-1H-pyrazolo[3,4-d]pyrimidine
 Methyl 2-hydroxy-4,6-dimethylpyrimidine-5-carboxylate Ethyl 2-hydroxy-4,6-dimethylpyrimidine-5-carboxylate Ethyl 2-chloro-4,6-dimethylpyrimidine-5-carboxylate 2-Chloro-4,6-dimethylpyrimidine-5-carboxylic acid
 Ethyl 4,6-dimethyl-2-methylthiopyrimidine-5-carboxylate Ethyl 2-amino-4,6-dimethylpyrimidine-5-carboxylate 2-Amino-4,6-dimethylpyrimidine-5-carboxylic acid Methyl 2-amino-4,6-dimethylpyrimidine-5-carboxylate
 2,6-Dichloro-4-hydroxypyrimidine 2-Ethyl-4,6-dihydroxypyrimidine 2-Ethyl-4,6-dichloropyrimidine Methyl 2,4-dichloro-6-methylpyrimidine-5-carboxylate
 4,4-Difluorocyclohexanone 3-Hydroxy-3-methylcyclobutanecarboxylic acid Methyl 4-methylnicotinate Ethyl 4-methylnicotinate
 3,3-Difluorocyclopentanecarboxylic acid 3-Bromopyrazolo[1,5-a]pyrimidine Ethyl pyrazolo[1,5-a]pyrimidine-3-carboxylate 2-Chloro-4-ethoxypyrimidine
 Ethyl 5-ethyl-6-hydroxy-2-methylpyrimidine-4-carboxylate Ethyl 6-chloro-5-ethyl-2-methylpyrimidine-4-carboxylate Ethyl 6-chloro-5-ethylpyrimidine-4-carboxylate Ethyl 6-hydroxy-5-ethylpyrimidine-4-carboxylate
 6-Hydroxy-5-methyl-2-(methylthio)pyrimidine-4-carboxylic acid (3,3-Difluorocyclopentyl)methanamine Methyl 3,3-difluorocyclopentanecarboxylate 2,4-Dimethoxy-5,6-dimethylpyrimidine
 2-Amino-6,7-dihydro-1H-cyclopenta[d]pyrimidin-4(5H)-one 2-Amino-4-chloro-6-(trifluoromethyl)pyrimidine 2-Methyl-4-amino-6-trifluoromethylpyrimidine Diisopropyl 3,3-dimethoxycyclobutane-1,1-dicarboxylate
 (1-(Aminomethyl)cyclobutyl)methanol 4-Bromo-3,5-difluoropyridine 7-Bromo-4-chloro-2-(methylthio)thieno[3,2-d]pyrimidine 2-Chloro-4-methylquinazoline
 4-Iodo-6-methoxypyrimidine 4-Hydroxy-6-(methylthio)pyrimido[5,4-d]pyrimidine 4-Chloro-2-(methylthio)-5,6,7,8-tetrahydroquinazoline 2-(Methylthio)-4-hydroxy-5,6,7,8-tetrahydroquinazoline
 4-Hydroxy-6-amino-5-(2,2-diethoxyethyl)-2-(methylthio)pyrimidine 2-Chloro-5-acetylpyrimidine 2-tert-Butyl-4-hydroxy-6-(trifluoromethyl)pyrimidine 4-Hydroxy-2-methoxy-6-(trifluoromethyl)pyrimidine
 4-Chloro-2-methoxy-6-(trifluoromethyl)pyrimidine 4-Hydroxy-6-amino-5-(2,2-dimethoxyethyl)-2-methylpyrimidine 4-Hydroxy-2-(methylthio)-7H-pyrrolo[2,3-d]pyrimidine 4-Hydroxy-2-methyl-7H-pyrrolo[2,3-d]pyrimidine
 4,6-Dimethyl-5-hydroxymethylpyrimidine 6-Chloro-4-amino-1-methylpyrazolo[4,5-e]pyrimidine 5-Chloro-6-iodopyridine-2,3-diamine N-(Phenylmethyl)-5-aminopyrimidine
 Methyl 4-amino-2-chloropyrimidine-5-carboxylate 4-Chloro-5-methyl-7H-pyrrolo[2,3-d]pyrimidine 1H-Indazole-3-methanol 5-(1-Aminoethyl)pyrimidine
 7-Chloro-[1,2,4]triazolo[1,5-c]pyrimidin-5-ol 5,7-Dichloro-[1,2,4]triazolo[1,5-c]pyrimidine 4,6-Dichloro-5-fluoro-2-methylpyrimidine 2-(Pyrrolidin-1-yl)pyrimidine-5-boronic acid pinacol ester
 2-(4-Boc-piperazin-1-yl)pyrimidine-5-boronic acid pinacol ester 2-(4-Methylpiperazin-1-yl)pyrimidine-5-boronic acid pinacol ester 2-Piperidinopyrimidine-5-boronic acid pinacol ester 2-(4-Morpholino)pyrimidine-5-boronic acid pinacol ester
 [2-[(tert-Butoxycarbonyl)amino]pyrimidin-5-yl]boronic acid pinacol ester 2-Methoxypyrimidine-5-boronic acid pinacol ester 2-Chloropyrimidine-5-boronic acid 4-(Aminomethyl)pyrimidine
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