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 Ethyl 5-bromo-2-methyl-3-indoleacetate ethyl 5-bromo-2-methoxybenzoate ethyl 5-bromo-2-ethylbenzoate ethyl 5-bromo-2-ethoxybenzoate
 ethyl 5-bromo-2,4-dimethylbenzoate ethyl 5-bromo-2,4-dimethoxybenzoate ethyl 5-bromo-2,4-diethoxybenzoate Ethyl 5-bromo-2,2-dimethyl-4-oxopentanoate
 ethyl 5-bromo-2-(trifluoromethoxy)benzoate ethyl 5-bromo-2-(piperidin-1-yl)benzoate ethyl 5-bromo-2-(dimethylamino)benzoate ethyl 5-bromo-2-(4-methylpiperazin-1-yl)benzoate
 Ethyl 5-bromo-1-methyl-1H-pyrazole-4-carboxylate Ethyl 5-bromo-1H-indole-2-carboxylate Ethyl 5-bromo-1H-indazole-3-carboxylate Ethyl 5-bromo-1,2,3-thiadiazole-4-carboxylate
 ethyl 5-bromo-1-(4-fluorophenyl)-1H-pyrazole-4-carboxylate ethyl 5-bromo-1-(3-chlorophenyl)-1H-pyrazole-4-carboxylate ethyl 5-bromo-1-(2-fluorophenyl)-1H-pyrazole-4-carboxylate Ethyl 5-benzyl-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridine-2-carboxylate
 Ethyl 5-aminothiazole-4-carboxylate Ethyl 5-Aminobenzofuran-2-Carboxylate ethyl 5-amino-4-phenylisoxazole-3-carboxylate ethyl 5-amino-4-cyano-3-methyl-2-thiophenecarboxylate
 Ethyl 5-amino-4-cyano-3-(2-ethoxy-2-oxoethyl)thiophene-2-carboxylate ethyl 5-amino-3-methylisothiazole-4-carboxylate Ethyl 5-amino-3-methyl-1H-pyrazole-4-carboxylate Ethyl 5-amino-2-pyrazinecarboxylate
 Ethyl 5-amino-2-methylthiazole-4-carboxylate Ethyl 5-amino-2-chlorobenzoate Ethyl 5-amino-1-tert-Butylpyrazole-4-carboxylate Ethyl 5-amino-1-phenyl-4-pyrazolecarboxylate
 Ethyl 5-amino-1-phenyl-1H-pyrazole-3-carboxylate Ethyl 5-amino-1-methyl-3-(trifluoromethyl)-1H-pyrazole-4-carboxylate Ethyl 5-amino-1-methyl-1H-pyrazole-4-carboxylate ethyl 5-amino-1H-pyrazole-4-carboxylate
 Ethyl 5-amino-1H-indazole-3-carboxylate ethyl 5-amino-1H-1,2,4-triazole-3-carboxylate ethyl 5-amino-1-ethyl-1H-pyrazole-4-carboxylate ethyl 5-amino-1-benzyl-1H-pyrazole-4-carboxylate
 Ethyl 5-amino-1,3,4-thiadiazole-2-carboxylate ethyl 5-amino-1,3,4-oxadiazole-2-carboxylate Ethyl 5-amino-1,2,3-thiadiazole-4-carboxylate ethyl 5-amino-1-(pyrimidin-2-yl)-1H-pyrazole-4-carboxylate
 ethyl 5-amino-1-(pyridin-4-yl)-1H-pyrazole-4-carboxylate ethyl 5-amino-1-(pyridin-2-yl)-1H-pyrazole-4-carboxylate ethyl 5-amino-1-(4-nitrophenyl)-1H-pyrazole-4-carboxylate Ethyl 5-amino-1-(4-methylphenyl)-1H-pyrazole-4-carboxylate
 Ethyl 5-amino-1-(4-fluorophenyl)-1H-pyrazole-4-carboxylate ethyl 5-amino-1-(4-bromophenyl)-1H-pyrazole-4-carboxylate ethyl 5-amino-1-(3-fluorophenyl)-1H-pyrazole-4-carboxylate Ethyl 5-amino-1-(3-chlorophenyl)-1H-pyrazole-4-carboxylate
 ethyl 5-amino-1-(2-fluorophenyl)-1H-pyrazole-4-carboxylate Ethyl 5-acetyloxyindole-2-carboxylate ethyl 5-acetylisoxazole-3-carboxylate Ethyl 5-[(4-N-Boc-amino)phenyl]-1,3-oxazole-4-carboxylate
 Ethyl 5,8-Dihydroxyimidazo[1,5-a]pyrazine-1-carboxylate Ethyl 5,8-Dichloroimidazo[1,5-a]pyrazine-1-carboxylate Ethyl 5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxylate ethyl 5,7-dichloropyrazolo[1,5-a]pyrimidine-3-carboxylate
 Ethyl 5,7-dichloro-1H-indole-2-carboxylate Ethyl 5,6-dimethyl-1H-benzimidazole-1-acetate Ethyl 5,6-dimethoxyindole-2-carboxylate Ethyl 5,6-dimethoxy-1H-indazole-3-carboxylate
 Ethyl 5,6-difluoro-1H-indazole-3-carboxylate Ethyl 5,6-dichloro-1H-indazole-3-carboxylate Ethyl 5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine-2-carboxylate ethyl 5,5-dimethyl-2,4-dioxohexanoate
 ethyl 5-(trifluoromethyl)-1-methyl-1H-pyrazole-4-carboxylate Ethyl 5-(trifluoromethyl)-1H-pyrazole-3-carboxylate Ethyl 5-(trifluoromethyl)-1H-indole-7-carboxylate ethyl 5-(trifluoromethyl)-1,2,4-oxadiazole-3-carboxylate
 ethyl 5-(trifluoromethyl)-1-(4-fluorophenyl)-1H-pyrazole-4-carboxylate Ethyl 5-(trifluoromethoxy)-1H-indole-2-carboxylate ethyl 5-(thiophen-2-yl)isoxazole-3-carboxylate Ethyl 5-(tert-butyl)-2H-pyrazole-3-carboxylate
 Ethyl 5-(Methylsulfonyl)pyridine-2-carboxylate ethyl 5-(hydroxymethyl)isoxazole-3-carboxylate ethyl 5-(chlorosulfonyl)-3-furoate ethyl 5-(chloromethyl)-3-isoxazolecarboxylate
 Ethyl 5-(chloromethyl)-2-furancarboxylate ethyl 5-(chloromethyl)-1,2,4-oxadiazole-3-carboxylate ethyl 5-(bromomethyl)thiazole-2-carboxylate ethyl 5-(aminomethyl)-2-furoate
 ethyl 5-(aminomethyl)-1,2,4-oxadiazole-3-carboxylate Ethyl 5-(5-bromo-2-thienyl)-3-isoxazolecarboxylate Ethyl 5-(4-nitrophenyl)oxazole-4-carboxylate ethyl 5-(4-methoxyphenyl)-1,2,4-oxadiazole-3-carboxylate
 Ethyl 5-(4-chlorophenyl)oxazole-4-carboxylate ethyl 5-(4-chlorophenyl)isoxazole-3-carboxylate Ethyl 5-(4-chlorophenyl)-2-formyl-3-furoate Ethyl 5-(4-chlorophenyl)-1,2,4-thiadiazole-3-carboxylate
 ethyl 5-(4-bromophenyl)isoxazole-3-carboxylate Ethyl 5-(4-bromophenyl)-1,3-oxazole-4-carboxylate Ethyl 5-(3-nitrophenyl)oxazole-4-carboxylate ethyl 5-(2-furyl)isoxazole-3-carboxylate
 ethyl 5-(2-furyl)-1-methyl-1H-pyrazole-3-carboxylate ethyl 5-(2-furyl)-1H-pyrazole-3-carboxylate ethyl 5-(2-chloroacetyl)-2,4-dimethyl-1H-pyrrole-3-carboxylate Ethyl 5-(2-bromoacetyl)isoxazole-3-carboxylate
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