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 3-benzyl-9-methyl-3,9-diazaspiro[5.5]undecane tert-butyl 9-methyl-3,9-diazaspiro[5.5]undecane-3-carboxylate 3-methyl-3,9-diazaspiro[5.5]undecane tert-butyl 3,9-diazaspiro[5.5]undecane-3-carboxylate
 2,4-dimethylthiophen-3-amine 2-methylbenzofuran (S)-(-)-1-Phenylethyl isocyanate (R)-(+)-1-Phenylethyl isocyanate
 4-((3-chloro-2,4-difluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate 4-chloro-7-methoxyquinazolin-6-yl acetate 4-((3-chloro-2,4-difluorophenyl)amino)-7-methoxyquinazolin-6-ol Ethyl 1-(aminomethyl)spiro[2.5]octane-1-carboxylate
 1-(((tert-butoxycarbonyl)amino)methyl)spiro[2.5]octane-1-carboxylic acid Ethyl 1-cyanospiro[2.5]octane-1-carboxylate Ethyl 2-cyano-2-cyclohexylideneacetate 1-(aminomethyl)spiro[2.5]octane-1-carboxylic acid
 1-(3-hydroxypropyl)-1H-benzo[d][1,2,3]triazole-5-carbaldehyde 1-(3-hydroxypropyl)-1H-benzo[d][1,2,3]triazole-5-carbonitrile 3-amino-4-((3-hydroxypropyl)amino)benzonitrile 4-((3-hydroxypropyl)amino)-3-nitrobenzonitrile
 1-(3-bromopropyl)-1H-benzo[d][1,2,3]triazole-5-carbaldehyde 8-[(R)-2-azido-1-(tert-butyl-dimethyl-silanyloxy)-ethyl]-5-benzyloxy-4H-benzo[1,4]oxazin-3-one (R)-8-(2-amino-1-((tert-butyldimethylsilyl)oxy)ethyl)-5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one (R)-8-(2-azido-1-hydroxyethyl)-5-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one
 (R)-8-(2-amino-1-hydroxyethyl)-5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one 8-(2-azidoacetyl)-5-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one 5-(benzyloxy)-8-(2-chloroacetyl)-2H-benzo[b][1,4]oxazin-3(4H)-one 8-acetyl-5-(benzyloxy)-2H-benzo[b][1,4]oxazin-3(4H)-one
 1-(3-amino-4-(benzyloxy)-2-hydroxyphenyl)ethanone 1-(4-(benzyloxy)-2-hydroxy-3-nitrophenyl)ethanone 1-(2,4-dihydroxy-3-nitrophenyl)ethanone 8-(2-aminoethyl)-5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one hydrochloride
 8-(2-aminoethyl)-5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one methyl 4-acetamido-5-iodo-2-methoxybenzoate (R)-5-(2-azido-1-((tert-butyldimethylsilyl)oxy)ethyl)-8-(benzyloxy)quinolin-2(1H)-one (R)-8-(benzyloxy)-5-(2-bromo-1-((tert-butyldimethylsilyl)oxy)ethyl)quinolin-2(1H)-one
 (R)-8-(benzyloxy)-5-(2-bromo-1-hydroxyethyl)quinolin-2(1H)-one Tert-butyl 3-oxo-1-oxa-4,9-diazaspiro[5.5]undecane-9-carboxylate Tert-butyl 4-(aminomethyl)-4-hydroxypiperidine-1-carboxylate Tert-butyl 1-oxa-6-azaspiro[2.5]octane-6-carboxylate
 Tert-butyl 1-oxa-4,9-diazaspiro[5.5]undecane-9-carboxylate 1-(2-methoxyphenyl)thiourea 4-methoxybenzo[d]thiazol-2-amine 4-methoxybenzo[d]thiazol-2(3H)-one
 7-acetyl-4-(benzyloxy)-1,3-benzothiazol-2(3H)-one 4-(benzyloxy)-7-(bromoacetyl)-1,3-benzothiazol-2(3H)-one 7-(2-azido-1-hydroxyethyl)-4-(benzyloxy)benzo[d]thiazol-2(3H)-one 7-[(1R)-2-azido-1-hydroxyethyl]-4-(benzyloxy)-1,3-benzothiazol-2(3H)-one
 (R)-7-(2-azido-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one 7-acetyl-4-methoxybenzo[d]thiazol-2(3H)-one 7-(2-bromoacetyl)-4-hydroxybenzo[d]thiazol-2(3H)-one N-(2-chloro-4-formyl-5-methoxyphenyl)acrylamide
 2-chloro-5-methoxyaniline 4-amino-5-chloro-2-methoxybenzaldehyde 2-isocyanato-1,1’-biphenyl Tert-butyl 2-hydroxy-7-azaspiro[3.5]nonane-7-carboxylate
 6-methoxyindoline 6-methoxyindoline-5-carbaldehyde Cis-tert-butyl 3,4-diazidopyrrolidine-1-carboxylate Cis-tert-butyl 3,4-dihydroxypyrrolidine-1-carboxylate
 GSK-961081; GSK-961081D; TD-5959; 961081; Batefenterol Succinate (R)-4-((3R,5R,8S,9S,10R,13R,14S,17R,E)-6-ethylidene-3-hydroxy-10,13-dimethyl-7-oxohexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanoic acid (R)-4-((3R,5S,8R,9S,10S,13R,14S,17R)-3-hydroxy-10,13-dimethyl-7-oxohexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanoic acid Obeticholic Acid;6-ECDCA; DSP-1747; INT-747
 3-(5-methyl-1H-pyrrol-3-yl)propanoic acid 3-(4-(ethoxycarbonyl)-5-methyl-1H-pyrrol-3-yl)propanoic acid Afatinib;Gilotrif;BIBW 2992;Tovok 4-bromo-1-chloro-2-(4-ethoxybenzyl)benzene
 (2S,3R,4S,5S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6,6-bis(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol (2S,3R,4S,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol Ertugliflozin; PF 04971729;MK-8835 Sitagliptin phosphate;Januvia;Glactiv;ONO-5435; MK-0431; L-000224715
 Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-3,4-dihydro-2H-pyran-3-yl)carbamate Tert-butyl ((1R,2S)-1-(2,5-difluorophenyl)-1-hydroxypent-4-yn-2-yl)carbamate Tert-butyl (1-(2,5-difluorophenyl)-1-oxopent-4-yn-2-yl)carbamate Tert-butyl (1-(methoxy(methyl)amino)-1-oxopent-4-yn-2-yl)carbamate
 2-((tert-butoxycarbonyl)amino)pent-4-ynoic acid Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-5-hydroxytetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2S,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2R,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
 Tert-butyl ((2S,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate Tert-butyl ((2R,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole benzenesulfonate 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole
 Tert-butyl 6a-hydroxy-1,2,6,6a-tetrahydropyrrolo[3,4-c]pyrazole-5(4H)-carboxylate (Z)-tert-butyl 3-((dimethylamino)methylene)-4-oxopyrrolidine-1-carboxylate Tert-butyl 2-(methylsulfonyl)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole 4-methylbenzenesulfonate
 Tert-butyl 4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate (2S,3R,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine AZD8186 PRT-060318;PRT318
 Omarigliptin;MK-3102 (R)-2-(2-methoxyphenyl)-2-((tetrahydro-2H-pyran-4-yl)oxy)ethanol BGB-324 BAR 502
 (S)-2-amino-3-(4-fluoro-1H-indol-3-yl)propanoic acid CMS-024; YSL; alpha-BCP[7-9];Tyroserleutide H3B-6527 BAR 501
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